Bophelo, Litokisetso
"Lantsid": litaelo bakeng sa ho sebelisoa, tlhaloso ya moriana, analogues, ulasan pelanggan
Liso tsa ka maleng ba lefu pampitšana tshilong ya dijo ka 'na la hlaha ka tšohanyetso. Bakeng sa ho phekoloa lefu lena lokela ho hang-hang a bale e gastroenterologist nang le phihlelo.
Ka mor'a ho hlahloba ka hloko ngaka lokelang ho hlalosa lithethefatsi-ba khahlanong le seso. The atlehang ka ho fetisisa ea bana ba lithethefatsi "Lantsid". Theko ea lithethefatsi ena tla ho tse thathamisitsoeng mona ka tlase. Ho phaella moo, u tla ithuta hore na thepa ke tlholeho ka o ile a re ho bolela, ha a ne a analogues efe kapa efe le kamoo ho ka nka hantle.
Sebopeho, tlhaloso, ambalaji le sebopeho
Ho lokisetsa "Lantsid" e ntshitsweng ka mokgwa wa capsules edible gelatin (thata). Ba na le 'mala o turquoise le dikahare ka mokgwa wa granules tšoeu.
The a sebetsang a motsoako ka lithethefatsi ena ke lansoprazole. Hape capsules e akarelletsa e latelang tšehetso likarolo: mannitol, povidone, lactose monohydrate, cetyl joala, sucrose le hypromellose phthalate.
O ne a nka meriana e rekiswa ho dipakete blister le mabokose.
phello ea moriana
ke lithethefatsi "Lantsid" ke efe? Litaelo bakeng sa ho sebelisoa e bolela hore ho ke ke sesitisa itseng tsa H + K + -ATPase (proton e pompo). metabolism lona e etsoa lisele tse (parietal) ea mpeng. Foromo ena le motho ea mafolofolo sulfonamide derivatives.
Sena se o beha diboloko moriana secretion ea acid e hydrochloric, fokotseha basal le susumelletseha secretion.
Ka lipophilicity phahameng, seo se bolela ho ena habonolo kenella ka hare ho lisele tse gastric (parietal), 'me joale, go tlhoma tlhaloganyo mo bona le fana ka le liphello tse cytoprotective, eketsa secretion ea bicarbonate le ho eketseha oxygenation ka sehloohong tshilong ya dijo lekala mucosa.
isa tekanyong le tekanyo ea thibelo ea basal le susumelletseha secretion ea acid e hydrochloric ba lethal dose-itšetlehileng ka eona. ph lona e ile ea eketseha ka mor'a lihora tse 1-2 le lihora tse 2-3 ka mor'a a e-ja ba mg, 15 of lithethefatsi le 30 ka ho latellana.
meriana ena ha e na le phello ho motility pampitšaneng ena gastrointestinal. Phello inhibitory ea lithethefatsi e ho bontšitsoe pele matsatsi a mane tsa baeti ba fihlelang ho. Mora phethoa kalafo bakeng sa lihora tse 40 acidity ntse bonyane 50% ya boemong ba basal.
a khaotsa ho tsuba ba ho lokisetsa joalo ha tloaelehileng.
thepa ya moriana
Ho lokisetsa "Lantsid" (letlapeng) ka mpeng mucosa liforomo IgA itseng bakeng sa Helicobacter pylori ke inhibiting kgolo ya H. pylori le ho eketseha mosebetsi oa meriana e meng.
Ho boetse ho bolela thibela tlhahiso ea pepsin le pepsinogen eketsa ea mahloriso maling.
The kinetics ya moriana
Hore na meriana e ananelang "Lantsid"? Litaelo bakeng sa ho sebelisoa e bolela hore absorption sena se bolela tshimolotse hang-hang ka mor'a ho lokisetsa siea le mala. Tlhōrō ea mahloriso ea lansoprazole ka mali ba ile ba hlokomela ka mor'a lihora tse 1,7.
tšebeliso lijo fokotsa absorption le bioavailability ya moriana.
The halofo bophelo ba lansoprazole ke lihora tse peli. Sena ha se ame bolelele ba hatelloang ea secretion gastric.
Qetello ea lithethefatsi 'meleng o etsoang tsoa le e bile le moroto.
ya litatoli na
Eo mafu a tsela e atlehang ka ho fetisisa itshwara moriana "Lantsid"? Reviews ba re ho ka sepheo se setle phekola mafu tse latelang:
- reflux esophagitis;
- bao e seng seso dyspepsia;
- lefu peptic seso (exacerbation) ya intestine le;
- esophagitis, erosive le ulcerative;
- liso tsa ka maleng oa khatello ea kelello e pampitšana tshilong ya dijo;
- Ellison - Zollinger.
Contraindications
Maemong a mang, u ke ke ua nka ho capsules "Lantsid"? Litaelo tsa Sebelisa e bolela hore contraindications ho nkoa ho bolela tse latelang boemo ba mokuli ha a re:
- kanyeso;
- trimester pele a bokhachane;
- lihlahala tse kotsi ka pampitšana tshilong ya dijo;
- Hypersensitivity ho dikarolo tsa moriana.
Ba qoaile lithethefatsi ena e hlophisitsweng bakeng sa batho ba nang le ho hloleha sebete, la bobeli le la boraro trimesters tsa boimana, bakuli ba hōlileng le bakuli ba sa reng letho ka.
Moriana o "Lantsid": litaelo tsa tšebeliso
Lohothwang komiki nkiloeng ka molomo. Ba lokela ho metsoa kaofela ntle ho hlafuna.
Ha erosive le ulcerative esophagitis le peptic seso tsa meriana mala balletsweng 30 mg, letsatsi le letsatsi bakeng sa dibeke tse 4-8. Haeba a lakatsa, litekanyetso li behoa ea ea eketseha ho 60 mg, ka ho ya ka letsatsi.
Ha liso khatello ea maikutlo le peptic lefu seso 12 duodenal seso meriana buelloa ho nka 30 mg, ka ho ya ka letsatsi le leng ka mohato o le mong. E etsa ka go tlhaolega hoseng, ka lijo tsa hoseng, tsa libeke tse 2-4.
The lefu Zollinger - Ellison meriana litekanyetso li behoa e fetola batho ka bomong.
Ha reflux esophagitis noa meriana nako e etsang khoeli ka palo ya mg, 30 ka letsatsi.
Ho felisa Helicobacter pylori lithethefatsi buelloa ho sebelisa 30 mg, habeli ka letsatsi. Ho ntlafatsa phekolo sephetho moriana o ho kopantswe le lithibela-mafu tse kang "clarithromycin" kapa "amoxicillin". Kalafo lokela ho nka bonyane beke.
Ka ulcerative dyspepsia ho lokisetsa e sebediswa bakeng sa ho libeke tse 2-4 ka lethal dose ea la 15-30 mg, ka ho ya ka letsatsi.
Ha sebete ho hloleha, hammoho le batho ba hōlileng ba qala phekolo le halofo lethal dose. Joale ba eketsehileng ho kgothaletswa, empa ho se ho feta 30 mg, ka ho ya ka letsatsi.
litla-morao
Moriana o "Lantsid Kit" ho ka etsa hore e itšoare ka e latelang-morao:
- hlooho e opang, ho tšoenyeha, malaise, ho otsela, ho tsekela, ho tepella maikutlo;
- fokotseha kapa ho eketsa ka takatso ea lijo, hyperbilirubinemia, ho nyekoa ke pelo, gastrointestinal candidiasis, bohloko mpeng, phahameng sebete transaminases, letšollo, ulcerative colitis, pipitlelano;
- khohlela, e ka holimo ho hema pampitšana tšoaetso ea, pharyngitis, ntaramane lefu, rhinitis;
- letlalo lekhopho, etymology multiforme, photosensitivity;
- khaello ea mali, thrombocytopenia;
- alopecia, myalgia.
ditshebeditsano lithethefatsi
Ho lokisetsa "Lantsid Kit", ae fokotsang lebelo mahlahana a ntsha tse metabolized ka sebete ka microsomal ho kena moea (mohlala, tse kang "Phenytoin" "Diazepam" le anticoagulants sa tobang).
Tshebediso tsoa hong ea lansoprazole, ae fokotsang lebelo le ph-itšetlehileng ka absorption ea lithethefatsi, bao e leng ea lihlopha tsa acid fokola. Hape nkoa moriana o eketsa absorption ea lithethefatsi tse lihlopha botlaaseng.
"Lantsid" thibela absorption "ketoconazole" tšepe letsoai "Ampicillin" le "Digoxin".
Lansoprazole ke 10% fokotsa rengwa "theophylline".
Sucralfate fokotsa bioavailability tsa lansoprazole ea 30%. Tabeng ena, ke habohlokoa ho boloka karohano pakeng tsa baeti ba fihlelang ho ea mokhoa oa itse (metsotso 30-40).
Lansoprazole e lumellana le "Indomethacin", "ibuprofen", "diazepam", "warfarin", "Propranolol" lithibela-pelehi molomo, hammoho le "prednisone" le "Phenytoin".
Antacids lokela ho tsamaisoa metsotso 60 pele kapa dihora tse 2 ka mor'a tsamaiso "Lantsida" hobane ba ne ba haholo fokotsa lebelo le ho fokotsa absorption ea bobeli.
likhothaletso itseng
Pele le ka mor'a phekolo le "Lantsid" hlokahalang endoscopic taolo ya boemo ba mokuli. Sena ke ho hlokahala hore ho busa tsoa ntshetsopeleng kankere, ka kalafo e ka pata matšoao a lefu lena le ho lieha ho fumanoe nepahetse.
Theko le analogues
Ke bokae ke "Lantsid" komiki? theko ea bona e ka bang 200 li-ruble. sesebelisoa sena se ka nka sebaka sa lithethefatsi tse ling haeba ho hlokahala. Ho etsa sena, a bua ka gastroenterologist ka.
Analogues ya moriana ka eona ke "Akrilanz", "Lansoprazole", "Gelikor", "Lanzaptor", "Lanzap", "Lanzabel", "Loenzar-Sanovel", "Lansofed", "Epicurus".
Reviews
bakuli ho fetisisa ho araba "Lantsid" lithethefatsi (analogs tsa lithethefatsi li ile tsa hlahisa ka holimo) feela ka lehlakoreng le nepahetseng. Bareki re ka mor'a matsatsi a 'maloa ea phekolo matšoao a sa thabiseng tsa lefu peptic seso hang-hang tsa nyamela. Ho feta moo, hammoho le meriana e meng sesebelisoa sa khothalletsa batho ka potlako ke pholiso erosions le ulceration ka mucosa ea intestine le.
The go tlhoka mesola ya meriana ena e kenyeletsa palo e khōlō ea liphetoho boima. Ha a ntse a mabapi le ditlhoko tsohle tsa ngaka tsa ponahalo ea bona ka ho qojoa.
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