Bophelo, Litokisetso
"Tolperisone" le bolela. Litaelo tsa tšebeliso
Tablets "Tolperisone" le akarelletsa sehlopha sa lithethefatsi, relaxants mesifa. The moriana o na le phello e bohareng. Lithethefatsi e na le lera botsitso mosebetsi, methapo ea kutlo-tšusumetso e tsoang ho, ae fokotsang lebelo le tiisetsa motoneurons le mathomo likhoele afferent. Sena se qholotsa emisang tsa poly- le monosynaptic reflexes lesapo la mokokotlo. Lithethefatsi thibela ho conduction ba nyakallo ka boko bakoang tsela reticulospinal. Ho sa tsotellehe hore sephetho sa tsamaiso ea methapo e bohareng e bolela ho eketseha pheriferale phallo ea mali. Ntshetsopeleng ya e le hantle ena e ka ba ka lebaka la tšusumetso ea antiadrenergicheskim le meriana antispasmodic. Ka ho sebelisa lithethefatsi ka molomo e hantle ananelang tswa intestine nyenyane. Ka mor'a halofo ea hora, ka hora lebetsoeng le hlokometse mahloriso palo e kahodimodimo ea lithethefatsi lero la mali. Ka lebaka persistemnogo bontša metabolism moriana o bioavailability ya 20%. The disintegration ea moriana o hlahellang teng liphio le sebete. Ka mokgwa wa metabolites ho 99% excreted ka moroto.
"Tolperisone" moriana. Litaelo ho sebelisoa. ya litatoli na
Abela sehlahisoa ka phahameng (pathologically) molumo le spasm ka mesifa striated amanang le bolwetse methapo ea kutlo manyolo ka diso tsa pampitšana pyramidal, setorouku, multiple sclerosis, encephalomyelitis, ho akarelletsa le myelopathy. The moriana o "Tolperisone" taeo pukwanana khothalletsa kalafo ka reductive mora tshebetso ka traumatology le malwetse a. Ke matšoao a kenyeletsa eketsehileng molumo le mesifa spasm, mesifa contracture, thatafatsa mafu tsamaisong ea musculoskeletal. Ka ho khetheha, ba lithethefatsi e atleha ho lumbar le bohloko cervical lefu, ramatiki ka manonyello kgolo, spondyloarthrosis, spondylosis. Hammoho le mekhoa e meng ea ba lokisetsa ho "Tolperisone 'kgothaletswa litaelo bakeng sa ho sebelisoa ho phekola occlusive vascular mofuta lefu.
"Tolperisone" meriana. Litaelo tsa tšebeliso
moriana o nkiloeng ka lethal dose ea pele ea 50 mg, ha ka makhetlo a fetang a mararo ka nako ya letsatsi. Butle-butle eketsa tjhelete ya etsoa lithethefatsi ho 150 mg, 2-3 leq. / Letsatsi la. nako e ikemiselitse ka bomong ho itšetlehile ka mofuta le ho tiea la puso lefu la mokuli.
Contraindications
Tablets "tolperisone" (likarabo tsa litsebi li tiisa hore) e sa abeloa ho masea a ka tlas'a ka ba lilemo li 18, ho se mamellane ea likarolo. Contraindications kenyeletsa ho ima le diabolololo. Ka lebaka la ho ba teng ha lactose ka meriana buelloa meriana mamellane kapa khaello ea ntho ena.
"Tolperisone" le bolela. Litaelo ho sebelisoa. liphetoho tse bohloko
moriana qholotsa hlooho, mesifa bofokoli, ho nyekoa ke pelo, gastralgia (matha ka litekanyetso li behoa tlaase). Ka lebaka la kalafo ea bonahala hypotension, alejiki itsoara joang ka bakoang ke ho se mamellane.
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