Bophelo, Litokisetso
Lithethefatsi "Lamikon": amohele taeo, ulasan pelanggan kopo, analogues, Sebopeho
Ke bokae ha lithethefatsi ena e le "Lamikon"? Theko ea lithethefatsi ena tla tšohloa sehloohong sena. Hape ho na le u tla fumana litaelo tse hlakileng tsa tšebeliso ea lithethefatsi, contraindications lona, analogs, ho bonahala, liphetoho e bohloko, foromo lokolloa, sebopeho le joalo-joalo.
Sebopeho, sebopeho le ambalaji tsa meriana
Fumana nkoa e le ea lithethefatsi e ka ba mefuta e latelang:
- "Lamikon" aerosol. Spray na le ntho a sebetsang a kang terbinafine. E le dikarolo tse eketsehileng tsa foromo ke propylene glycol, macrogol cetostearyl phenylate 20, acid e benzoic, disodium edetate, le metsi bakeng sa ente Poloxamer 407. epicutaneous lithethefatsi e lokolloa ka botlolo e nang le pompo metering ka 25 g.
- Cream "Lamikon" (mafura). Motataisi o tlaleha hore karolo ea mafolofolo foromo ena boetse eo sebeletsa terbinafine. metsoako tse ling tsa mofuta ona li: diminerale oli, hydroxide sodium, tšoeu bonolo parafini, cetostearyl joala le phenylethyl, macrogol cetostearyl phenylate 20, propylene glycol, poloxamer 407 ba le metsi a hloekisitsoeng. Ka rekisa mafura bo fihla ka methapo ea 15 g,
- "Lamikon" molomo lokisetsa. Tablets, thuto eo e kenyeleditsweng ka lebokoseng entsoe ka lebokoso, hape e na le e joalo e ntho a sebetsang a ke terbinafine. Mabapi le dikarolo tse eketsehileng, ba ile ba kenyelletsa: poone starch, sodium starch glycolate, microcrystalline selulose, colloidal anhydrous silica, hydroxypropylmethylcellulose le magnesium stearate. matlapa a fumanoang liseleng tsa ea moeli ea likotoana 7.
pharmacodynamics
Diokobatsi sehlopha nkoa lithethefatsi - antifungal. Ho ea ka litaelo tseo, ka motsoako o ka sehloohong oa moemeli ena ke alilamin eo hlahisa e sebetsang phekolo phello palo e khōlō ea mefuta e fapaneng li-fungus.
The fungicidal thepa ea terbinafine (tloaelehile mahloriso) le ho aba ka dermatophyte li-fungus, hammoho le mefuta e meng ea li-fungus dimorphic.
Ho itšetlehile ka mofuta, le tomoso moriana hona ka 'na ea bontša bobeli fungicidal le fungistatic mosebetsi.
Molao-motheo oa ho sebetsa
Joang lithethefatsi "Lamikon"? Tataiso e tlaleha hore moemeli ena ka ho toba thibela ho ba sethaleng pele tsa sterol biosynthesis ka lera la seleng e fungal. Le ka lebaka la ho pepesehela joalo a amoheleha intracellular bokella squalene, 'me ho hloka ergosterol. Sena se etsa hore ho timetsoa ha lisele tse fungal.
The mochine ea nkang khato ea chelete le ka ho toba e amanang le ho tshebetso ya ho thibelo ya potlakisang tsebetso ea lik'hemik'hale squalene epoxidase joaloka, e amana le cytochrome P-450.
Ho ea ka litsebi, lithethefatsi "Lamikon" ha e na tšusumetso e ka liphello tsa lithethefatsi tse ling, 'me ka metabolism hormonal.
Pharmacokinetics
E le lithethefatsi e ananelang, "Lamikon"? Tataiso e bolela hore ha sebakeng seo kapa lihlooho tsa puisano kopo absorption ea lithethefatsi a sebetsang a ke ka tlase ho 5% ea lethal dose ea sebelisoa. Ka lebaka leo, ho pepesehela lona systemic e tlaase.
Ha laolwa ka lihlooho lithethefatsi hang-hang o qala ho ba le phello e le ke haholo e atlehang bakeng sa nako e khutšoanyane (hoo e ka bang 8-13 matsatsi).
Ka ho boloka ea mahloriso a lakatsa ya moriana ka stratum corneum tsa epidermis, e leng ile a fumana ka nako ya phekolo, ketso fungicidal ya moriana o le e tsoela pele ka beke e 'ngoe ka mor'a khanselwa lona.
Ha ke tlosoa ka molomo, "Lamikona" ntho a sebetsang a bakoang ke ho letlalo la, manala le moriri. Ea mahloriso ea lithethefatsi dinama tse nyenyane tse ka ka ho feletseng e fana ka thepa ea lona fungicidal.
Absorption matlapa a 70%, mme bioavailability bona e feletseng - 50%.
Ba ile ba fumana paakanyong ka palo ea 250 mg, ke mahloriso phahameng ka ho fetisisa ea mali e ka mor'a hora halofo. E atlehang halofo bophelo nakong ka 30 lihora tse.
Lijo e hanyenyane feela ama bioavailability ya moriana. Le protheine lero la mali e tlama ho ntho mafolofolo 99,5%. Meriana ena ka potlako le kenella ka hare ho dermis le bakoang ka stratum corneum.
Ho itšehla thajana "Lamikona" etsoang ke litsoelesa le sebaceous. Hape, e fumanoa moriri, letlalo le moriri follicles. Ka libeke tse ea pele ea phekolo, lithethefatsi le kenella ka hare ho poleiti Nail.
Terbinafine e metabolized kapele le cytochrome P 450. Ka mor'a biotransformation sehlahisoa nkiloeng metabolites khathetseng moeeng ke liphio.
Ha ntho e sa tloaelehang ka sebete 'me liphio rengwa terbinafine lebelo, ae fokotsang lebelo haholo, ho etsa hore ea mahloriso e phahameng ka lero la mali.
ho bonahala
Ho tloha nakong eo a khethe liforomo ea moo litekanyetso li behoa "Lamikon" lithethefatsi? Setlolo, litaelo bakeng sa tšebeliso eo e hlalosoa mona ka tlase, hammoho le ho fafatsa le na le matšoao a latelang:
- diso fungal letlalo, tse neng di le bakoang ke li-fungus ba genus Trichophyton, Microsporum le Epidermophyton (maoto a dermotofitiya, groin, 'mele, joalo-joalo);
- multicolor (kapa pityriasis) versicolor, eo a tsoa ho tswa ho sephetho sa Malassezia li-fungus;
- candidiasis tsa letlalo, e leng e ile ea tsosa ke li-fungus ba genus Candida.
Ka morero ofe sebelisoa liforomo tsa molomo "Lamikon" (matlapa) ya moriana? Tataiso e tlaleha matšoao tse latelang:
- tsoaetsanang fungal tsa letlalo, moo ata bona, mahloriso kapa ho hlahisa maikutlo a joalo e le hore ba lokela ho tšoaroa hantle ho tsela molomo (feela rerang Ngaka e);
- mycosis hlooho le onychomycosis (tsoaetsanang Nail lipoleiti).
Re lokela ho hlokomela hore "Lamikon" matlapa a ha sebelisoa bakeng sa ho phekoloa 'mala (kapa scaly) zoster.
Contraindications
Mofuta ofe contraindications lokela ho hlokomela tsa pele o sebelisa lithethefatsi "Lamikon"? Motataisi o ile a re feela thibelong e feletseng ea mefuta eohle ea meriana e nkoa hypersensitivity ho ntho lona.
Ha e le nako ea boimana, bongoaneng le anyesa, ba contraindications e lekanyelitsoeng.
Mafura "Lamikon": litaelo tsa tšebeliso
liforomo tse joalo tsa lithethefatsi, e le spray le le mafura, o fana ka maikutlo a kopo bona kantle. Pele li sebelisa bakeng sa ho phekoloa mafu a fungal, o lokela ho pele hloekileng le omella ho libakeng tse amehang ea letlalo.
Ho itšetlehile ka ho tiea ha lefu lena le mofuta oa pathogen lithethefatsi "Lamikon" (mafura) sebelisoa habeli ka letsatsi. Aerosol e sebediswa le maqhubu a tšoanang.
tranelate le lokela ho ho sebediswa eseng feela hore le e amehang ea letlalo fungus e, empa e boetse e le libakeng tse bapileng. Ho phetha mokhoa ona ke ho hotle ho lera tšesaane butle-butle hohla mafura likoahelo.
Ha mafu a tšoaetsanoang e tsamaea leleire lekhopho (mohlala, tlas'a matsoele, groin, maraong kapa pakeng tsa menoana), le libakeng tse tšoaroa lokela ho koahela gauze (bosiu).
Tshebediso ya aerosol
Ke lokela ho sebedisa Spray "Lamikon"? profesionalce Reviews tlaleha hore e le sebelisitsoe ka palo e lekaneng ea ho moisten ka ho fafatsa ka libakeng tse le ho ba hlolloa ha le li-fungus, hammoho le letlalo ka bophelo bo botle le haufi le eona.
Ka nako ea phekolo e itšetlehile ka mecha ea litaba ea moo lefu tiea (ho fihlela ho libeke tse peli).
Setšoantšo sa mokuli o ile a hlokomela ka matsatsi a 'maloa. Bakeng sa kalafo e atlehang haholoanyane, ho hlokahala hore ba khomarele litaelo ka tieo ho se hopotse kopo e mong 'me a sa ho emisa kalafo pele ho nako. Ho seng joalo ho na le ke kotsing e khōlō ea ho oela ketsong ena hape.
Tsela ea ho nka matlapa ao?
Diokobatsi sehlopha hore owns meriana ka pel'a rōna, o ile a bontša ka ditaelo. O re bolella ka tsela eo ho etsa sesebelisoa seo.
E le busa, "Lamikon" lipilisi laetsoeng ho bana ho tloha le lilemo li 6, hammoho le bakuli ba batho ba baholo. Fumana ho lokisetsa molomo e tsoela pele ho fihlela ho nyamela ka ho feletseng le matšoao 'ohle a lefu le fungal (ho itšetlehile ka mofuta le ho tiea).
The litšila tsa litekanyetso li behoa moriana o bakeng sa batho ba baholo ke 250 mg,, le bakeng sa bana ba bekha 20-40 lik'hilograma - 125 mg,. Le boima ba 'mele e khōlō ea ngoana e le tseo ke li behetsoeng 250 mg, ea moriana.
Ka nako ea phekolo le trichophytosis le letlalo candidosis ke libeke tse 2-4, 'me ka Tinea pedis - libeke tse 2-6.
mafu Fungal la hlooho ho ka tloaelehileng bana. E le busa, ba ile ba ba amenable ho kalafo ha moriana le sebelisitsoe ka dosages ea kgothaletswa ke ngaka e etsang khoeli.
Onychomycosis kalafo nka libeke tse 6 bakeng sa manala le 12 - bakeng sa monoana Nail. Tlas'a fokotswa kgolo ya Nail lipoleiti phekolo ka nako e telele.
liphetoho tse bohloko
Local lithethefatsi "Lamikon", analogues ya tse ho tse thathamisitsoeng ka tlaase mona, li ka etsa hore matšoao a kang letlalo gommage, tukang, ho hlohlona, ho utloa bohloko, ho teneha, pigmentation phytoteratology, etymology le karolong e ka holimo le thehoa. Ba ka boela ba fumana kulisa.
Ha fumana matlapa a, tse latelang litla rateheng:
- neutropenia, agranulocytosis, Lyell lefu, pancytopenia, Stevens-Johnson lefu;
- thrombocytopenia, liphetoho anaphylactoid, meferefere tatso, matšoao a lupus, hlooho;
- photosensitivity, paresthesia, hypoesthesia, neuralgia;
- ho tsekela, boikutlo ba ho ba botlalo ka mpeng, letšollo, ho lahleheloa ke takatso ea lijo;
- exacerbation ea psoriasis, ho nyekoa ke pelo, psoriasiform rashes, bohloko mpeng, myalgia;
- urticaria, arthralgia, lekhopho, generalized pustulosis, tahlehelo moriri, keketseho ea enzyme sebete;
- mokhathala, hepatobiliary ho se sebetse, nyooko, lefu la sebete.
Analogs le theko ea lithethefatsi e
Ke bokae sethethefatsi "Lamikon"? Theko ea lithethefatsi ena e itšetlehile ka sebopeho lona. Mafura le fafatsa ka rekoa bakeng sa li-ruble 180-220, 'me matlapa a - bakeng sa 370-400 li-ruble.
Ha e le counterparts, har'a atlehang haholoanyane o ka abelwang karolo ya chelete tse kang "Amorolak" acid e salicylic. "Mikoseptin", "Nitrofungin", "Mikolak", "Exoderil".
Reviews of moriana o
Feedback ho ba 'nile ba sebelisa lithethefatsi "Lamikon" ba-positive, haholo. Bakuli ba tlaleha hore phekolo bohlokwa ba tsamaiso ea lithethefatsi ena e se e ile a re matsatsi a 'maloa ka mor'a tšebeliso a hae a sebetsang. Ka tloaelo ho, lefu le fungal le disappears ho ea qetellong ea tsela ea phekolo.
Maemong a matla, lingaka nkhothaletsa hlakanywa litekanyetso li behoa foromo (mohlala, matlapa a le mafura, fafatsa le matlapa).
Ho phaella ho melaetsa tse ntle mabapi le "Lamikon" ho lokisetsa ea mo khahlanyetsa 'me poeletsotlaleho negative. Ba ba atisa ho amahanngoa le katleho ha eona. Leha ho le joalo, litsebi li bolela hore sena se ka etsahala feela ka kalafo ya bao e seng hlokolosi ho li-fungus moriana o kapa sebelisoa hampe. Ka hona, pele ho sebelisa setlolo, matlapa kapa spray buelloa ho bona ngaka le ho theha moemeli causative tsa mafu a fungal.
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